Enzyme Inhibitors

Blocking Peptides Decrease Tissue Transglutaminase Processing of Gliadin in Vitro

Engineering / Fluorescence / Enzyme Inhibitors / In Vitro / Gliadin / Animals / Peptides / Agricultural / CHEMICAL SCIENCES / Enzyme activity / Agricultural and Food Chemistry / Amino Acid Sequence / Tissue Transglutaminase / Transglutaminases / Molecular Sequence Data / Animals / Peptides / Agricultural / CHEMICAL SCIENCES / Enzyme activity / Agricultural and Food Chemistry / Amino Acid Sequence / Tissue Transglutaminase / Transglutaminases / Molecular Sequence Data

Blocking Peptides Decrease Tissue Transglutaminase Processing of Gliadin in Vitro

Engineering / Fluorescence / Enzyme Inhibitors / In Vitro / Gliadin / Animals / Peptides / Agricultural / CHEMICAL SCIENCES / Enzyme activity / Agricultural and Food Chemistry / Amino Acid Sequence / Tissue Transglutaminase / Transglutaminases / Molecular Sequence Data / Animals / Peptides / Agricultural / CHEMICAL SCIENCES / Enzyme activity / Agricultural and Food Chemistry / Amino Acid Sequence / Tissue Transglutaminase / Transglutaminases / Molecular Sequence Data

Blocking Peptides Decrease Tissue Transglutaminase Processing of Gliadin in Vitro

Engineering / Fluorescence / Enzyme Inhibitors / In Vitro / Gliadin / Animals / Peptides / Agricultural / CHEMICAL SCIENCES / Enzyme activity / Agricultural and Food Chemistry / Amino Acid Sequence / Tissue Transglutaminase / Transglutaminases / Molecular Sequence Data / Animals / Peptides / Agricultural / CHEMICAL SCIENCES / Enzyme activity / Agricultural and Food Chemistry / Amino Acid Sequence / Tissue Transglutaminase / Transglutaminases / Molecular Sequence Data

Blocking Peptides Decrease Tissue Transglutaminase Processing of Gliadin in Vitro

Engineering / Fluorescence / Enzyme Inhibitors / In Vitro / Gliadin / Animals / Peptides / Agricultural / CHEMICAL SCIENCES / Enzyme activity / Agricultural and Food Chemistry / Amino Acid Sequence / Tissue Transglutaminase / Transglutaminases / Molecular Sequence Data / Animals / Peptides / Agricultural / CHEMICAL SCIENCES / Enzyme activity / Agricultural and Food Chemistry / Amino Acid Sequence / Tissue Transglutaminase / Transglutaminases / Molecular Sequence Data

Phosphoramidate Dinucleosides as Hepatitis C Virus Polymerase Inhibitors

Organic Chemistry / Medicinal Chemistry / Modeling / Enzyme Inhibitors / Magnetic Resonance Spectroscopy / In Vitro / Humans / Virus / Hepatitis C Virus / Organophosphorus Compounds / Medicinal / Molecular Model / Nucleosides / Chemical Synthesis / Oxidation-Reduction / In Vitro / Humans / Virus / Hepatitis C Virus / Organophosphorus Compounds / Medicinal / Molecular Model / Nucleosides / Chemical Synthesis / Oxidation-Reduction

Glucosidase Inhibitory Anthranols, Kenganthranols A−C, from the Stem Bark of Harungana m adagascariensis

Natural Products / Cameroon / Enzyme Inhibitors / Medicinal Plants / Biological Sciences / Saccharomyces cerevisiae / CHEMICAL SCIENCES / Anthraquinones / Natural / Saccharomyces cerevisiae / CHEMICAL SCIENCES / Anthraquinones / Natural

Quinoxalinylurea derivatives as a novel class of JSP-1 inhibitors

Organic Chemistry / Enzyme Inhibitors / Computer Model / Urea / Structure activity Relationship / Protein Tyrosine Phosphatases / Dual Specificity Phosphatases / Protein Tyrosine Phosphatases / Dual Specificity Phosphatases

Quinoxalinylurea Derivatives as a Novel Class of JSP-1 Inhibitors

Organic Chemistry / Enzyme Inhibitors / Computer Model / Urea / Structure activity Relationship / Protein Tyrosine Phosphatases / Dual Specificity Phosphatases / Protein Tyrosine Phosphatases / Dual Specificity Phosphatases

UDP-galactose 4-epimerase from Kluyveromyces fragilis

Biochemistry / Protein Folding / Catalysis / Kinetics / Mass Spectrometry / Enzyme Inhibitors / Urea / Sodium Dodecyl Sulfate-Polyacrylamide Gel Electrophoresis / Enzyme / High Pressure Liquid Chromatography / European / Monomer / Substrate Specificity / Amino Acid Profile / Molecular weight / Amino Acid Sequence / Quntitative Thin Layer Chromatography / Protein Binding / Protein Denaturation / Ligands / Chemical Modification / Biochemistry and cell biology / Dimerization / Molecular Sequence Data / Enzyme Inhibitors / Urea / Sodium Dodecyl Sulfate-Polyacrylamide Gel Electrophoresis / Enzyme / High Pressure Liquid Chromatography / European / Monomer / Substrate Specificity / Amino Acid Profile / Molecular weight / Amino Acid Sequence / Quntitative Thin Layer Chromatography / Protein Binding / Protein Denaturation / Ligands / Chemical Modification / Biochemistry and cell biology / Dimerization / Molecular Sequence Data

Nebivolol Increases Arterial Distensibility In Vivo

Enzyme Inhibitors / Cardiovascular Risk / Hypertension / Hemodynamics / Sheep / Blood Pressure / Nitric oxide / Animals / Arterial stiffness / Clinical Sciences / Nitric Oxide Synthase / Pulse Wave Velocity / Nitroglycerin / Vascular Resistance / Atenolol / Blood Pressure / Nitric oxide / Animals / Arterial stiffness / Clinical Sciences / Nitric Oxide Synthase / Pulse Wave Velocity / Nitroglycerin / Vascular Resistance / Atenolol

Nebivolol Increases Arterial Distensibility In Vivo

Enzyme Inhibitors / Cardiovascular Risk / Hypertension / Hemodynamics / Sheep / Blood Pressure / Nitric oxide / Animals / Arterial stiffness / Clinical Sciences / Nitric Oxide Synthase / Pulse Wave Velocity / Nitroglycerin / Vascular Resistance / Atenolol / Blood Pressure / Nitric oxide / Animals / Arterial stiffness / Clinical Sciences / Nitric Oxide Synthase / Pulse Wave Velocity / Nitroglycerin / Vascular Resistance / Atenolol

Sarco-endoplasmic reticulum Ca2+ ATPase (SERCA) inhibitors identify a novel calcium pool in the central nervous system

Neurochemistry / Calcium / Enzyme Inhibitors / Magnesium / ATPase / Permeability / Animals / Male / Endoplasmic Reticulum / Central Nervous System / Neurons / Astrocytes / Rats / Rat / Wistar Rats / Ion Transport / Brain Chemistry / Neurosciences / Sarcoplasmic reticulum / Permeability / Animals / Male / Endoplasmic Reticulum / Central Nervous System / Neurons / Astrocytes / Rats / Rat / Wistar Rats / Ion Transport / Brain Chemistry / Neurosciences / Sarcoplasmic reticulum

Structure-based inhibitor design of AccD5, an essential acyl-CoA carboxylase carboxyltransferase domain of Mycobacterium tuberculosis

Computational Biology / Kinetics / Enzyme Inhibitors / Multidisciplinary / Antibiotic Resistance / Crystal structure / Tuberculosis / Mycobacterium tuberculosis / Escherichia coli / Drug Design / Active site / Substrate Specificity / Fatty Acid / National Cancer Institute / University of Southern California / Cell Wall / In Silico / Protein Quaternary Structure / Ligands / Crystal structure / Tuberculosis / Mycobacterium tuberculosis / Escherichia coli / Drug Design / Active site / Substrate Specificity / Fatty Acid / National Cancer Institute / University of Southern California / Cell Wall / In Silico / Protein Quaternary Structure / Ligands

Phenoxyacetohydrazide Schiff bases: β-Glucuronidase inhibitors

Organic Chemistry / Enzyme Inhibitors / Animals / Glucuronidase / Schiff bases / Cattle / Molecules / Cattle / Molecules

A novel thermostable neutral proteinase from Saccharomonospora canescens

Kinetics / Fluorescence / Calcium / Enzyme Inhibitors / Sequence Analysis / Biological Sciences / Physical sciences / Temperature / Activation Energy / Zinc / Enzyme / Actinomycetales / Substrate Specificity / Molecular Mass / Atomic Absorption / Esterases / Energy Transfer / Amino Acid Sequence / Polyacrylamide Gel Electrophoresis / Protein Binding / Chelating Agents / Hydrogen-Ion Concentration / Melting Temperature / Proteolytic activity / Molecular Sequence Data / Biological Sciences / Physical sciences / Temperature / Activation Energy / Zinc / Enzyme / Actinomycetales / Substrate Specificity / Molecular Mass / Atomic Absorption / Esterases / Energy Transfer / Amino Acid Sequence / Polyacrylamide Gel Electrophoresis / Protein Binding / Chelating Agents / Hydrogen-Ion Concentration / Melting Temperature / Proteolytic activity / Molecular Sequence Data

O exercício físico atenua o déficit autonômico cardíaco induzido pelo bloqueio da síntese do óxido nítrico

Enzyme Inhibitors / Autonomic Nervous System / Hypertension / Blood Pressure / Animals / Male / Heart rate / Rats / Nitric Oxide Synthase / Analysis of Variance / Wistar Rats / Propranolol / Arquivos brasileiros / Male / Heart rate / Rats / Nitric Oxide Synthase / Analysis of Variance / Wistar Rats / Propranolol / Arquivos brasileiros
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